Endothelin-1 vs Leuphasyl

Head-to-head comparison of Endothelin-1 (Endothelin-1) and Leuphasyl (Pentapeptide-18) — benefits, dosing, side effects, research data, and where to buy.

Research Score

PropertyEndothelin-1Leuphasyl
CategorySkin & CosmeticSkin & Cosmetic
Full NameEndothelin-1Pentapeptide-18
Molecular Weight2493 Da569.6 Da
Half-Life~2–10 minutesN/A
Amino Acids215
Typical Dose1–100 nM0.01-2% in cosmetic formulations
RouteIn vitro / ex vivoTopical
Purity≥98%≥98%
Studies Count35022
Research StatusPre-clinicalClinical

Endothelin-1 Benefits

  • Stimulates melanocyte activity
  • Supports melanosome transfer studies
  • Useful in UV-induced pigmentation research
  • Links vascular and pigment signaling

Leuphasyl Benefits

  • wrinkle-appearance reduction
  • expression-line softening
  • topical anti-aging support
  • cosmetic skin-smoothing

Endothelin-1 Dosing

1 nM exposure|10 nM exposure|100 nM exposure

Leuphasyl Dosing

Topical serum/cream 0.01-2%|Apply once or twice daily|Combine with moisturizer or peptide serum

Endothelin-1 Side Effects

  • Vasoconstriction
  • Cell-stress signaling at high concentrations
  • Inflammatory cross-talk

Leuphasyl Side Effects

  • temporary redness
  • mild irritation
  • sensitivity in compromised skin

Research Overview

Endothelin-1

Endothelin-1 is one of the best-studied non-melanocortin regulators of pigmentation in human skin. It is strongly associated with UV-induced tanning responses and pigment disorder biology.

Leuphasyl

Pentapeptide-18 has published cosmetic and formulation literature supporting its use in anti-aging skincare. Evidence is strongest for topical cosmetic smoothing rather than deep structural remodeling.

Ready to buy?

Find both peptides from our verified, lab-tested vendors with purity certificates and third-party testing.

Common Stacking Partners

Endothelin-1 stacks with:

ACTHL-tyrosine

Leuphasyl stacks with:

RetinoidsHyaluronic AcidPeptide Complexes
endothelinpigmentationmelanocyteuv-responseanti-wrinkletopicalpeptideexpression-lines