AICAR vs Neuropeptide S

Head-to-head comparison of AICAR (5-Aminoimidazole-4-carboxamide Ribonucleotide (Acadesine)) and Neuropeptide S (Neuropeptide S) — benefits, dosing, side effects, research data, and where to buy.

Research Score

PropertyAICARNeuropeptide S
CategoryPerformanceCognitive Enhancement
Full Name5-Aminoimidazole-4-carboxamide Ribonucleotide (Acadesine)Neuropeptide S
Molecular Weight338.21 g/mol2203 Da
Half-Life~2-3 hoursMinutes to <1 hour
Amino AcidsNucleoside analog20
Typical DoseResearch-only; no validated human dose
RouteIntracerebroventricular/Intranasal
Purity>99%≥98%
Studies Count18028
Research StatusActive ResearchPre-clinical

AICAR Benefits

  • Increases endurance capacity, enhances fatty acid oxidation, promotes mitochondrial biogenesis, improves glucose uptake, cardioprotective effects

Neuropeptide S Benefits

  • anxiolysis
  • stress resilience
  • attention support
  • arousal modulation

AICAR Dosing

Research doses: 50-150 mg subcutaneously. Typically administered 30-60 minutes before physical activity in research settings.

Neuropeptide S Dosing

0.1-1 nmol i.c.v. in animal studies|intranasal research-only exploration|no established human protocol

AICAR Side Effects

  • Potential hypoglycemia, lactic acidosis at high doses, injection site reactions. Banned by WADA as a metabolic modulator.

Neuropeptide S Side Effects

  • sleep disruption
  • headache
  • jitteriness

Research Overview

AICAR

Salk Institute researchers demonstrated AICAR could increase endurance in sedentary mice by 44% without exercise training. Activates AMPK, triggering PGC-1α expression, mitochondrial biogenesis, and enhanced fatty acid β-oxidation.

Neuropeptide S

Animal studies suggest NPS can reduce anxiety-like behavior while altering wakefulness and alertness through the NPS receptor system. Human cognitive data are very limited, and it has no approved clinical indication.

Ready to buy?

Find both peptides from our verified, lab-tested vendors with purity certificates and third-party testing.

Common Stacking Partners

AICAR stacks with:

MOTS-cGW501516

Neuropeptide S stacks with:

BromantaneTianeptine sodium
AMPK-activatorenduranceexercise-mimeticfat-oxidationcardioprotectivepeptideanxiolyticstress