Synthetic PeptidesClinical
Cilengitide
Cilengitide cyclic RGD pentapeptide integrin antagonist
Amino Acids
N/A
Molecular Weight
N/A
Half-life
N/A
Research Score
4.7
Studies
92
Storage
Store lyophilized at -20°C, reconstituted at 2-8°C
What is Cilengitide?
A synthetic cyclic peptide containing the RGD motif that antagonizes integrins alpha-v-beta-3 and alpha-v-beta-5. It was advanced clinically as an antiangiogenic and antitumor agent.
Key Benefits & Mechanisms
Integrin antagonist
Anticancer
Macrocyclic peptide
Research Summary
Research