Tianeptine sodium vs Macimorelin

Head-to-head comparison of Tianeptine sodium (Tianeptine sodium) and Macimorelin (Macimorelin acetate (AEZS-130)) — benefits, dosing, side effects, research data, and where to buy.

PropertyTianeptine sodiumMacimorelin
CategoryCognitive EnhancementGrowth Hormone
Full NameTianeptine sodiumMacimorelin acetate (AEZS-130)
Molecular Weight458.94 DaN/A
Half-LifeAbout 2.5 hoursabout 4-6 hours
Amino AcidsN/AN/A
Typical Dose12.5 mg 3 times daily0.5 mg/kg single oral dose
RouteOralOral
Purity≥98%≥98%
Studies Count280120
Research StatusClinicalClinical

Tianeptine sodium Benefits

  • mood improvement
  • anxiety reduction
  • cognitive clarity
  • stress adaptation

Macimorelin Benefits

  • diagnostic GH stimulation
  • single oral dose
  • rapid measurable GH response
  • high clinical utility

Tianeptine sodium Dosing

12.5 mg oral 3x/day|25 mg/day oral|clinical antidepressant dosing

Macimorelin Dosing

0.5 mg/kg orally as a single dose|fasted testing conditions|serial GH sampling after administration

Tianeptine sodium Side Effects

  • nausea
  • dizziness
  • dependence risk

Macimorelin Side Effects

  • dysgeusia or taste disturbance
  • nausea
  • headache

Research Overview

Tianeptine sodium

Clinical studies support tianeptine as an antidepressant with a distinctive glutamatergic and neuroplasticity-related profile. Some evidence suggests cognitive benefits in mood-impaired populations, likely secondary to improved stress handling and affect.

Macimorelin

Macimorelin has been validated in clinical testing as an oral alternative to injectable GH stimulation tests. Its short-term use makes it a useful translational tool for evaluating pituitary GH reserve.

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Common Stacking Partners

Tianeptine sodium stacks with:

BromantanePRL-8-53

Macimorelin stacks with:

Pituitary testingEndocrine workup
antidepressantanxiolyticmooddiagnosticghrelin-mimeticgh-stimulation-test