Tesofensine vs L-692,429

Head-to-head comparison of Tesofensine (Tesofensine (NS2330)) and L-692,429 (L-692,429) — benefits, dosing, side effects, research data, and where to buy.

Research Score

PropertyTesofensineL-692,429
CategoryWeight ManagementGrowth Hormone
Full NameTesofensine (NS2330)L-692,429
Molecular Weight426.52 g/molN/A
Half-Life~200-300 hoursunknown / study-dependent
Amino AcidsSmall moleculeN/A
Typical Dose0.03-0.1 mg/kg
RouteOral
Purity>98%≥98%
Studies Count3530
Research StatusPhase III Clinical TrialsPre-clinical

Tesofensine Benefits

  • Potent appetite suppression, increased metabolic rate, enhanced thermogenesis, improved mood during dieting, reduces food reward-seeking behavior

L-692,429 Benefits

  • potent GHSR agonism
  • oral bioactivity in models
  • validates ghrelin pathway
  • useful research probe

Tesofensine Dosing

Clinical doses: 0.25-1.0 mg orally once daily. Research typically uses 0.5 mg. Extremely long half-life (8-13 days) means steady-state in 7-10 days.

L-692,429 Dosing

0.03-0.1 mg/kg in early studies|single oral or short-course research dosing|serial GH sampling recommended

Tesofensine Side Effects

  • Dry mouth, insomnia, constipation, increased heart rate, elevated blood pressure. Not recommended with uncontrolled hypertension.

L-692,429 Side Effects

  • increased appetite
  • glucose intolerance
  • transient prolactin changes

Research Overview

Tesofensine

Phase II trials showed 12.8 kg average weight loss at 1.0 mg dose over 6 months. Simultaneously inhibits reuptake of norepinephrine, dopamine, and serotonin, producing appetite suppression and increased thermogenesis.

L-692,429

L-692,429 was important in early GH secretagogue research because it showed that nonpeptide molecules could trigger robust GH release. It remains a classic tool compound for studying receptor-mediated GH pulsatility and appetite signaling.

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Common Stacking Partners

Tesofensine stacks with:

5-Amino-1MQAOD-9604MOTS-c

L-692,429 stacks with:

Receptor assaysEndocrine studies
weight-lossappetite-suppressanttriple-reuptake-inhibitorthermogenesistool-compoundgh-secretagogueghrelin-pathway