Neuropeptide S vs Macimorelin

Head-to-head comparison of Neuropeptide S (Neuropeptide S) and Macimorelin (Macimorelin acetate (AEZS-130)) — benefits, dosing, side effects, research data, and where to buy.

Research Score

PropertyNeuropeptide SMacimorelin
CategoryCognitive EnhancementGrowth Hormone
Full NameNeuropeptide SMacimorelin acetate (AEZS-130)
Molecular Weight2203 DaN/A
Half-LifeMinutes to <1 hourabout 4-6 hours
Amino Acids20N/A
Typical DoseResearch-only; no validated human dose0.5 mg/kg single oral dose
RouteIntracerebroventricular/IntranasalOral
Purity≥98%≥98%
Studies Count28120
Research StatusPre-clinicalClinical

Neuropeptide S Benefits

  • anxiolysis
  • stress resilience
  • attention support
  • arousal modulation

Macimorelin Benefits

  • diagnostic GH stimulation
  • single oral dose
  • rapid measurable GH response
  • high clinical utility

Neuropeptide S Dosing

0.1-1 nmol i.c.v. in animal studies|intranasal research-only exploration|no established human protocol

Macimorelin Dosing

0.5 mg/kg orally as a single dose|fasted testing conditions|serial GH sampling after administration

Neuropeptide S Side Effects

  • sleep disruption
  • headache
  • jitteriness

Macimorelin Side Effects

  • dysgeusia or taste disturbance
  • nausea
  • headache

Research Overview

Neuropeptide S

Animal studies suggest NPS can reduce anxiety-like behavior while altering wakefulness and alertness through the NPS receptor system. Human cognitive data are very limited, and it has no approved clinical indication.

Macimorelin

Macimorelin has been validated in clinical testing as an oral alternative to injectable GH stimulation tests. Its short-term use makes it a useful translational tool for evaluating pituitary GH reserve.

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Common Stacking Partners

Neuropeptide S stacks with:

BromantaneTianeptine sodium

Macimorelin stacks with:

Pituitary testingEndocrine workup
peptideanxiolyticstressdiagnosticghrelin-mimeticgh-stimulation-test