Nafarelin vs Cetrorelix

Head-to-head comparison of Nafarelin (Nafarelin acetate) and Cetrorelix (Cetrorelix acetate) — benefits, dosing, side effects, research data, and where to buy.

Research Score

PropertyNafarelinCetrorelix
CategorySexual HealthSexual Health
Full NameNafarelin acetateCetrorelix acetate
Molecular Weight1321.47 Da1431.06 Da
Half-Life~2-4 hours~30 hours
Amino Acids1010
Typical Dose200 mcg intranasal twice daily0.25 mg SC daily
RouteIntranasalSubcutaneous
Purity≥98%≥98%
Studies Count220300
Research StatusClinicalClinical

Nafarelin Benefits

  • pituitary suppression
  • cycle scheduling
  • endometriosis-related reproductive care
  • controlled hormone modulation

Cetrorelix Benefits

  • prevents premature ovulation
  • supports IVF cycle control
  • blocks LH surge
  • short-acting pituitary suppression

Nafarelin Dosing

200 mcg intranasal twice daily|0.4 mg/day intranasal|protocol-based suppression cycles

Cetrorelix Dosing

0.25 mg SC daily|start on stimulation day 5-6|protocol-dependent antagonist cycle

Nafarelin Side Effects

  • nasal irritation
  • hot flashes
  • headache

Cetrorelix Side Effects

  • injection-site reactions
  • headache
  • nausea

Research Overview

Nafarelin

Nafarelin has a long history in reproductive medicine, especially for endometriosis and cycle suppression. Studies show it down-regulates the HPG axis after an initial stimulatory flare.

Cetrorelix

Cetrorelix is a cornerstone GnRH antagonist in assisted reproduction, with a fast onset and reversible suppression of LH. Trials show it improves cycle management by reducing premature ovulation during stimulation.

Ready to buy?

Find both peptides from our verified, lab-tested vendors with purity certificates and third-party testing.

Common Stacking Partners

Nafarelin stacks with:

FSHhCG

Cetrorelix stacks with:

FSHhCG
GnRH-agonistfertilityendocrinologyGnRH-antagonistivf