Met-enkephalin vs Teduglutide

Head-to-head comparison of Met-enkephalin (Tyr-Gly-Gly-Phe-Met) and Teduglutide (Teduglutide (glycyl-2 human glucagon-like peptide-2 analog)) — benefits, dosing, side effects, research data, and where to buy.

Research Score

PropertyMet-enkephalinTeduglutide
CategoryPain ManagementGastrointestinal
Full NameTyr-Gly-Gly-Phe-MetTeduglutide (glycyl-2 human glucagon-like peptide-2 analog)
Molecular Weight573.67 Da3752 Da
Half-Life1-5 minutes in plasmaapproximately 2-3 hours
Amino Acids533
Typical Dose0.1-5 ug per animal0.05 mg/kg/day
RouteIntrathecal / intracerebroventricularSubcutaneous
Purity≥98%≥98%
Studies Count1200300
Research StatusPre-clinicalClinical

Met-enkephalin Benefits

  • endogenous opioid signaling
  • analgesic reference ligand
  • spinal antinociception
  • neurochemical pain-pathway probe

Teduglutide Benefits

  • mucosal-growth
  • absorption-support
  • barrier-repair
  • intestinal-adaptation

Met-enkephalin Dosing

Intrathecal 0.1-5 ug per animal|Intracerebroventricular 0.1-2 ug per animal|In vitro 1-100 nM

Teduglutide Dosing

0.05 mg/kg once daily subcutaneous injection|chronic maintenance dosing in approved use|monitor fluid status and intestinal anatomy

Met-enkephalin Side Effects

  • sedation at higher exposure
  • constipation-like opioid effects
  • rapid enzymatic degradation

Teduglutide Side Effects

  • abdominal pain
  • fluid retention
  • polyp/neoplasia monitoring needed

Research Overview

Met-enkephalin

Met-enkephalin has been extensively used in receptor pharmacology and nociception studies to map mu and delta opioid biology. The main limitation in translational work is very short half-life from peptidase cleavage and poor systemic stability.

Teduglutide

Teduglutide has robust clinical evidence showing improved intestinal absorption and reduced parenteral nutrition dependence in short bowel syndrome. Its mechanism, via GLP-2 receptor activation, makes it highly relevant to mucosal healing and intestinal adaptation research.

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Common Stacking Partners

Met-enkephalin stacks with:

gabapentinketamine

Teduglutide stacks with:

nutritional-supportoral-rehydrationprobiotics
opioid-peptideenkephalinmu-opioidanalgesiashort-bowelmucosal-healingabsorptionintestinal-adaptationGLP-2