Cosyntropin vs Macimorelin

Head-to-head comparison of Cosyntropin (Cosyntropin (ACTH 1-24)) and Macimorelin (Macimorelin acetate (AEZS-130)) — benefits, dosing, side effects, research data, and where to buy.

Research Score

PropertyCosyntropinMacimorelin
CategoryPain ManagementGrowth Hormone
Full NameCosyntropin (ACTH 1-24)Macimorelin acetate (AEZS-130)
Molecular Weight2933.3 DaN/A
Half-Life~10 minabout 4-6 hours
Amino Acids24N/A
Typical Dose0.25 mg IV/IM diagnostic dose|off-label headache protocols vary0.5 mg/kg single oral dose
RouteIV|IMOral
Purity≥98%≥98%
Studies Count61120
Research StatusClinical researchClinical

Cosyntropin Benefits

  • refractory migraine
  • anti-inflammatory signaling
  • headache rescue research

Macimorelin Benefits

  • diagnostic GH stimulation
  • single oral dose
  • rapid measurable GH response
  • high clinical utility

Cosyntropin Dosing

0.25 mg IV/IM|1 mg IV/IM

Macimorelin Dosing

0.5 mg/kg orally as a single dose|fasted testing conditions|serial GH sampling after administration

Cosyntropin Side Effects

  • flushing
  • nausea

Macimorelin Side Effects

  • dysgeusia or taste disturbance
  • nausea
  • headache

Research Overview

Cosyntropin

Cosyntropin is not a standard pain drug, but it appears in headache literature because ACTH analogs can help some patients with difficult migraine attacks. The analgesic rationale is partly tied to steroidogenic and anti-inflammatory effects.

Macimorelin

Macimorelin has been validated in clinical testing as an oral alternative to injectable GH stimulation tests. Its short-term use makes it a useful translational tool for evaluating pituitary GH reserve.

Ready to buy?

Find both peptides from our verified, lab-tested vendors with purity certificates and third-party testing.

Common Stacking Partners

Cosyntropin stacks with:

ACTH(1-24)Synacthen

Macimorelin stacks with:

Pituitary testingEndocrine workup
migraineheadacheACTH-analogdiagnosticghrelin-mimeticgh-stimulation-test