Buserelin vs Cetrorelix

Head-to-head comparison of Buserelin (Buserelin acetate) and Cetrorelix (Cetrorelix acetate) — benefits, dosing, side effects, research data, and where to buy.

Research Score

PropertyBuserelinCetrorelix
CategorySexual HealthSexual Health
Full NameBuserelin acetateCetrorelix acetate
Molecular Weight1239.39 Da1431.06 Da
Half-Life~50-80 minutes~30 hours
Amino Acids910
Typical Dose200 mcg intranasal 3x daily|0.2-0.5 mg SC daily|depot per protocol0.25 mg SC daily
RouteIntranasal/SubcutaneousSubcutaneous
Purity≥98%≥98%
Studies Count450300
Research StatusClinicalClinical

Buserelin Benefits

  • pituitary down-regulation
  • cycle synchronization
  • ovarian stimulation control
  • fertility protocol timing

Cetrorelix Benefits

  • prevents premature ovulation
  • supports IVF cycle control
  • blocks LH surge
  • short-acting pituitary suppression

Buserelin Dosing

200 mcg intranasal 3x daily|0.2-0.5 mg SC daily|depot injection per protocol

Cetrorelix Dosing

0.25 mg SC daily|start on stimulation day 5-6|protocol-dependent antagonist cycle

Buserelin Side Effects

  • hot flashes
  • headache
  • initial LH/FSH flare

Cetrorelix Side Effects

  • injection-site reactions
  • headache
  • nausea

Research Overview

Buserelin

Buserelin has been studied extensively as a GnRH agonist in IVF down-regulation and other reproductive-endocrine protocols. Its use helped establish modern cycle-control approaches in assisted reproduction.

Cetrorelix

Cetrorelix is a cornerstone GnRH antagonist in assisted reproduction, with a fast onset and reversible suppression of LH. Trials show it improves cycle management by reducing premature ovulation during stimulation.

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Common Stacking Partners

Buserelin stacks with:

FSHhCG

Cetrorelix stacks with:

FSHhCG
GnRH-agonistfertilityivfGnRH-antagonist