Cetrorelix vs Nafarelin

Head-to-head comparison of Cetrorelix (Cetrorelix acetate) and Nafarelin (Nafarelin acetate) — benefits, dosing, side effects, research data, and where to buy.

Research Score

PropertyCetrorelixNafarelin
CategorySexual HealthSexual Health
Full NameCetrorelix acetateNafarelin acetate
Molecular Weight1431.06 Da1321.47 Da
Half-Life~30 hours~2-4 hours
Amino Acids1010
Typical Dose0.25 mg SC daily200 mcg intranasal twice daily
RouteSubcutaneousIntranasal
Purity≥98%≥98%
Studies Count300220
Research StatusClinicalClinical

Cetrorelix Benefits

  • prevents premature ovulation
  • supports IVF cycle control
  • blocks LH surge
  • short-acting pituitary suppression

Nafarelin Benefits

  • pituitary suppression
  • cycle scheduling
  • endometriosis-related reproductive care
  • controlled hormone modulation

Cetrorelix Dosing

0.25 mg SC daily|start on stimulation day 5-6|protocol-dependent antagonist cycle

Nafarelin Dosing

200 mcg intranasal twice daily|0.4 mg/day intranasal|protocol-based suppression cycles

Cetrorelix Side Effects

  • injection-site reactions
  • headache
  • nausea

Nafarelin Side Effects

  • nasal irritation
  • hot flashes
  • headache

Research Overview

Cetrorelix

Cetrorelix is a cornerstone GnRH antagonist in assisted reproduction, with a fast onset and reversible suppression of LH. Trials show it improves cycle management by reducing premature ovulation during stimulation.

Nafarelin

Nafarelin has a long history in reproductive medicine, especially for endometriosis and cycle suppression. Studies show it down-regulates the HPG axis after an initial stimulatory flare.

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Common Stacking Partners

Cetrorelix stacks with:

FSHhCG

Nafarelin stacks with:

FSHhCG
GnRH-antagonistfertilityivfGnRH-agonistendocrinology