AICAR vs DSIP

Head-to-head comparison of AICAR (5-Aminoimidazole-4-carboxamide Ribonucleotide (Acadesine)) and DSIP (Delta Sleep-Inducing Peptide) — benefits, dosing, side effects, research data, and where to buy.

Research Score

PropertyAICARDSIP
CategoryPerformancePerformance
Full Name5-Aminoimidazole-4-carboxamide Ribonucleotide (Acadesine)Delta Sleep-Inducing Peptide
Molecular Weight338.21 g/mol848.8 Da
Half-Life~2-3 hours~15-25 minutes
Amino AcidsNucleoside analog9
Typical Dose100-200 mcg
RouteSC / IV / Intranasal
Purity>99%
Studies Count18074
Research StatusActive ResearchPre-clinical

AICAR Benefits

  • Increases endurance capacity, enhances fatty acid oxidation, promotes mitochondrial biogenesis, improves glucose uptake, cardioprotective effects

DSIP Benefits

  • Promotes deep delta wave sleep
  • Normalizes disrupted sleep patterns
  • Reduces cortisol and stress response
  • Pain modulating effects
  • Antioxidant properties

AICAR Dosing

Research doses: 50-150 mg subcutaneously. Typically administered 30-60 minutes before physical activity in research settings.

DSIP Dosing

Standard: 100-200 mcg SC or IV, 30-60 min before bed|Cycle: 10-14 days, 5-7 days off|Chronic insomnia: 100 mcg daily for 2-3 weeks|Can be combined with Ipamorelin pre-bed

AICAR Side Effects

  • Potential hypoglycemia, lactic acidosis at high doses, injection site reactions. Banned by WADA as a metabolic modulator.

DSIP Side Effects

  • Common (Mild): Morning grogginess initially, mild headache
  • Rare: Vivid dreams, temporary appetite changes
  • Generally very well tolerated

Research Overview

AICAR

Salk Institute researchers demonstrated AICAR could increase endurance in sedentary mice by 44% without exercise training. Activates AMPK, triggering PGC-1α expression, mitochondrial biogenesis, and enhanced fatty acid β-oxidation.

DSIP

DSIP has moderate clinical evidence from European studies. Human trials show improved sleep quality and normalized sleep-wake cycles. Also studied for alcohol and opiate withdrawal. Unique mechanism distinct from traditional sleep aids.

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Common Stacking Partners

AICAR stacks with:

MOTS-cGW501516

DSIP stacks with:

IpamorelinSelankEpithalon
AMPK-activatorenduranceexercise-mimeticfat-oxidationcardioprotectiveSleepStress ReliefRecoveryPerformance