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MetabolicPre-clinical

Adipotide

CKGGRAKDC-GG-D(KLAKLAK)2 (Fat Cell Targeting)

Amino Acids

N/A

Molecular Weight

~2,500 Da

Half-life

~hours (estimated)

Research Score

3.5

Studies

12

Storage

N/A

What is Adipotide?

Adipotide is a peptidomimetic that targets and destroys the blood supply to fat tissue (adipose vasculature). It uses a homing sequence to find blood vessels feeding white fat cells and a proapoptotic sequence to destroy them. Studied for rapid, targeted fat loss in primate models.

Key Benefits & Mechanisms

Targeted fat cell destruction

Rapid fat loss in primate studies

Selective for white adipose tissue

Does not affect other tissues

Significant weight reduction in animal models

Unique mechanism of action

Potential for spot reduction

Research Summary

Adipotide showed dramatic fat loss results in rhesus monkeys (11% body weight in 4 weeks). However, renal toxicity was observed, limiting clinical development. The concept of vascular targeting for fat reduction is novel. Significant safety hurdles remain before human use.