Histatin-5 vs Macimorelin

Head-to-head comparison of Histatin-5 (Human histatin 5) and Macimorelin (Macimorelin acetate (AEZS-130)) — benefits, dosing, side effects, research data, and where to buy.

Research Score

PropertyHistatin-5Macimorelin
CategoryDental & OralGrowth Hormone
Full NameHuman histatin 5Macimorelin acetate (AEZS-130)
Molecular Weight3035 DaN/A
Half-Lifeminutes in salivaabout 4-6 hours
Amino Acids24N/A
Typical Dose1-100 µM in research formulations0.5 mg/kg single oral dose
RouteTopical/Oral rinseOral
Purity≥98%≥98%
Studies Count120120
Research StatusPre-clinicalClinical

Histatin-5 Benefits

  • anti-Candida activity
  • biofilm suppression
  • mucosal wound support
  • oral innate immunity

Macimorelin Benefits

  • diagnostic GH stimulation
  • single oral dose
  • rapid measurable GH response
  • high clinical utility

Histatin-5 Dosing

topical rinse or gel|short contact exposure|repeat applications in research protocols

Macimorelin Dosing

0.5 mg/kg orally as a single dose|fasted testing conditions|serial GH sampling after administration

Histatin-5 Side Effects

  • local irritation
  • proteolytic instability
  • dose-dependent cytotoxicity in vitro

Macimorelin Side Effects

  • dysgeusia or taste disturbance
  • nausea
  • headache

Research Overview

Histatin-5

Histatin-5 is a major salivary defense peptide that can kill Candida species and influence oral microbial communities. It is also investigated for wound-healing and xerostomia-associated oral infection models.

Macimorelin

Macimorelin has been validated in clinical testing as an oral alternative to injectable GH stimulation tests. Its short-term use makes it a useful translational tool for evaluating pituitary GH reserve.

Ready to buy?

Find both peptides from our verified, lab-tested vendors with purity certificates and third-party testing.

Common Stacking Partners

Histatin-5 stacks with:

chlorhexidinefluoridexylitol

Macimorelin stacks with:

Pituitary testingEndocrine workup
antimicrobial-peptidecandidasalivaoral-defensediagnosticghrelin-mimeticgh-stimulation-test